We are one of the most trusted exporters, suppliers, and traders, of Prilocaine Injection in various sterile packaging options. The offered injection is used as intermediate-acting local anesthetic in various tasks of dentistry. It is formulated for injection use and contains Prilocaine HCL as the active ingredient. Prilocaine Injection is also used widely for intravenous regional anaesthesia as it safely and effectively numbs the area for performing the surgery. It effects the local anesthetic action by stabilizing the neuronal membrane that inhibits the ionic fluxes required for the initiation and conduction of impulses.
Sterile, non-pyrogenic isotonic solution
Administered by infiltration or by nerve block
Low cardiac toxicity
Typically NLT 98%
Used as a local anaesthetic and is often used in dentistry.
Prilocaine binds to the intracellular surface of sodium channels which blocks the subsequent influx of sodium into the cell. Action potential propagation and never function is, therefore, prevented. This block is reversible and when the drug diffuses away from the cell, sodium channel function is restored and nerve propagation returns.
Mode of Action:
Prilocaine acts on sodium channels on the neuronal cell membrane, limiting the spread of seizure activity and reducing seizure propagation. The antiarrhythmic actions are mediated through effects on sodium channels in Purkinje fibers.
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